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Found 5 of ec50 data for polymerid = 6577
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50236535(CHEMBL1231132)
Affinity DataEC50:  80nMAssay Description:Inhibition of PDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM227594(PS10)
Affinity DataEC50:  456nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged SUMO-fused PDK2 expressed in Escherichia coli BL-21 cells preincubated for 15 mins followed by...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50525863(CHEMBL1708524)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of PDK2 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50525865(CHEMBL1419854)
Affinity DataEC50:  3.80E+3nMAssay Description:Inhibition of PDK2 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50525864(CHEMBL1733274)
Affinity DataEC50:  5.20E+3nMAssay Description:Inhibition of PDK2 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed