Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Inhibition of PDK2 (unknown origin)More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 456nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged SUMO-fused PDK2 expressed in Escherichia coli BL-21 cells preincubated for 15 mins followed by...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Inhibition of PDK2 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 3.80E+3nMAssay Description:Inhibition of PDK2 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Capital Medical University
Curated by ChEMBL
Capital Medical University
Curated by ChEMBL
Affinity DataEC50: 5.20E+3nMAssay Description:Inhibition of PDK2 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair